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STD1T
CAS No. 893075-58-6
STD1T( USP2a inhibitor STD1T )
Catalog No. M16439 CAS No. 893075-58-6
STD1T (USP2a inhibitor STD1T) is a hit-to-lead, small-molecule inhibitor of USP2a with IC50 of 3.3 uM in Ub-AMC assays.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 598 | Get Quote |
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| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameSTD1T
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NoteResearch use only, not for human use.
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Brief DescriptionSTD1T (USP2a inhibitor STD1T) is a hit-to-lead, small-molecule inhibitor of USP2a with IC50 of 3.3 uM in Ub-AMC assays.
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DescriptionSTD1T (USP2a inhibitor STD1T) is a hit-to-lead, small-molecule inhibitor of USP2a with IC50 of 3.3 uM in Ub-AMC assays, displays no activity against USP7 at 10 uM.
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In VitroSTD1T inhibits USP2a enzymatic activity in a concentration dependent manner. STD1T shows selective inhibition of USP2a vs. USP7 at the concentrations of 10 μM and 2000 μM, respectively.
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In Vivo——
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SynonymsUSP2a inhibitor STD1T
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PathwayProteasome/Ubiquitin
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TargetDUB
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RecptorDUB
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Research Area——
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Indication——
Chemical Information
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CAS Number893075-58-6
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Formula Weight417.498
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Molecular FormulaC19H19N3O4S2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 62.5 mg/mL (149.70 mM)
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SMILESO=C(C1=C(NC(COCC2=NOC(C3=CC=CS3)=C2)=O)SC4=C1CCCC4)N
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Chemical Name2-(2-((5-(thiophen-2-yl)isoxazol-3-yl)methoxy)acetamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Tomala MD, et al. Eur J Med Chem. 2018 Apr 25;150:261-267.
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