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VU534

CAS No. 923509-20-0

VU534( —— )

Catalog No. M36972 CAS No. 923509-20-0

VU534 is a NAPE-PLD agonist with an EC50 of 0.30 μM.VU534 is a dual inhibitor of FAAH and sEH, with an IC50 of 1.2 μM for sEH.VU534 is used in diseases related to cardiometabolism.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

VU534
Note

Research use only, not for human use.
Brief Description

VU534 is a NAPE-PLD agonist with an EC50 of 0.30 μM.VU534 is a dual inhibitor of FAAH and sEH, with an IC50 of 1.2 μM for sEH.VU534 is used in diseases related to cardiometabolism.
Description

VU534 is a NAPE-PLD activator, with an EC50 of 0.30 μM. VU534 is dual inhibitors of FAAH and sEH (IC50 of 1.2 μM). VU534 increases efferocytosis in a NAPE-PLD dependent manner. VU534 has the potential for cardiometabolic diseases study .
In Vitro

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In Vivo

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Synonyms

——
Pathway

Metabolic Enzyme/Protease
Target

FAAH
Recptor

FAAH | Phospholipase | Epoxide Hydrolase
Research Area

——
Indication

——

Chemical Information

CAS Number

923509-20-0
Formula Weight

447.55
Molecular Formula

C21H22FN3O3S2
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 25 mg/mL (55.86 mM; Ultrasonic )
SMILES

CC1=CC2=C(SC(NC(=O)C3CCN(CC3)S(=O)(=O)C3=CC=C(F)C=C3)=N2)C(C)=C1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Jonah E Zarrow, et al. Small Molecule Activation of NAPE-PLD Enhances Efferocytosis by Macrophages. ACS Chem. Biol. 2023, 18, 8, 1891–1904. ?

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