Org 25543
CAS No. 363628-88-0
Org 25543( —— )
Catalog No. M28443 CAS No. 363628-88-0
Org 25543 is the development of an N-Acyl amino acid that selectively inhibits the glycine transporter 2 to produce analgesia in a rat model of chronic pain.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 131 | In Stock |
|
| 5MG | 117 | In Stock |
|
| 10MG | 174 | In Stock |
|
| 25MG | 290 | In Stock |
|
| 50MG | 384 | In Stock |
|
| 100MG | 539 | In Stock |
|
| 200MG | 710 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameOrg 25543
-
NoteResearch use only, not for human use.
-
Brief DescriptionOrg 25543 is the development of an N-Acyl amino acid that selectively inhibits the glycine transporter 2 to produce analgesia in a rat model of chronic pain.
-
DescriptionOrg 25543 is the development of an N-Acyl amino acid that selectively inhibits the glycine transporter 2 to produce analgesia in a rat model of chronic pain.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayMembrane Transporter/Ion Channel
-
TargetChloride Channel
-
RecptorCRTh2 (DP2) receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number363628-88-0
-
Formula Weight412.53
-
Molecular FormulaC24H32N2O4
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCOc1cc(cc(OC)c1OCc1ccccc1)C(=O)NCC1(CCCC1)N(C)C
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
-
Anestan
Halothane is an inhalational general anesthetic. It is the only inhalational anesthetic containing bromine.
-
DCPIB
DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μM, demonstrating at least 100-fold higher affinity over TREK1/TRAAK channels.?DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC), has been reported to activate TREK1 and TREK2 in astrocytes and in vitro recently.?
-
VU 0240551
VU 0240551 is a potent, selecticve inhibitor of the neuronal K-Cl cotransporter KCC2 with IC50 of 568 nM in K+ uptake assay in KCC2-overexpressing cells.
Cart
sales@molnova.com