Desketoraloxifene

CAS No. 216570-81-9

Desketoraloxifene( —— )

Catalog No. M23980 CAS No. 216570-81-9

Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 272 In Stock
10MG 409 In Stock
25MG 737 In Stock
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Biological Information

  • Product Name
    Desketoraloxifene
  • Note
    Research use only, not for human use.
  • Brief Description
    Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).
  • Description
    Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Phospholipase
  • Recptor
    PLD1|PLD2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    216570-81-9
  • Formula Weight
    445.57
  • Molecular Formula
    C27H27NO3S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C1CCN(CC1)CCOC2=CC=C(C=C2)C3=C(SC4=C3C=CC(=C4)O)C5=CC=C(C=C5)O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Scott S A , Spencer C T , MC O’Reilly, et al. Discovery of Desketoraloxifene Analogues as Inhibitorsof Mammalian, Pseudomonas aeruginosa, and NAPE PhospholipaseD Enzymes[J]. Acs Chemical Biology, 2015, 10(2):421.
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