Cart
sales@molnova.com
LSD1-IN-7 benzenesulfonate
CAS No. 2097523-60-7
LSD1-IN-7 benzenesulfonate( CC-90011 benzenesulfonate )
Catalog No. M23947 CAS No. 2097523-60-7
LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 170 | In Stock |
|
| 2MG | 74 | In Stock |
|
| 5MG | 120 | In Stock |
|
| 10MG | 188 | In Stock |
|
| 25MG | 330 | In Stock |
|
| 50MG | 479 | In Stock |
|
| 100MG | 695 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameLSD1-IN-7 benzenesulfonate
-
NoteResearch use only, not for human use.
-
Brief DescriptionLSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
-
DescriptionLSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
-
In Vitro——
-
In VivoAnimal Model:BALB/c nude mice bearing small cell lung carcinoma (SCLC)Dosage:5 mg/kg Administration:Oral administration; daily; for 30 days Result:Showed a tumor growth inhibition (TGI) of 78% at 5 mg/kg with nobody weight loss.
-
SynonymsCC-90011 benzenesulfonate
-
PathwayChromatin/Epigenetic
-
TargetHistone Demethylase
-
RecptorLSD1
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2097523-60-7
-
Formula Weight609.64
-
Molecular FormulaC30H29F2N5O5S
-
Purity>98% (HPLC)
-
SolubilityDMSO:60mg/ml(98.42mM; Need ultrasonic)
-
SMILESN#CC1=CC=C(C(N=C(N2CCC(N)CC2)N3C)=C(C4=CC=C(OC)C(F)=C4)C3=O)C=C1F.O=S(C5=CC=CC=C5)(O)=O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Young K. Chen, et al. Compositions comprising an inhibitor of lysine specific demethylase-1. WO2017079670A1.
molnova catalog
related products
-
GSK-2879552
A potent, selective irreversible inhibitor of LSD1 with Ki app of 1.7 uM.
-
KDM4C-IN-1
KDM4C-IN-1 is a selective and potent KDM4C inhibitor (IC50: 8 nM) with potential anticancer activity.KDM4C-IN-1 inhibits the growth of HepG2 and A549 cells, and can be used for the study of leukaemia.
-
E67-2
E67-2 is a potent and selective inhibitor of H3K9 Jumonji demethylase KIAA1718 (KDM7A) with IC50 of 3.4 uM.
