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Home - Products - Chromatin/Epigenetic - Histone Demethylase - LSD1-IN-7 benzenesulfonate

LSD1-IN-7 benzenesulfonate

CAS No. 2097523-60-7

LSD1-IN-7 benzenesulfonate( CC-90011 benzenesulfonate )

Catalog No. M23947 CAS No. 2097523-60-7

LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 170 In Stock
2MG 74 In Stock
5MG 120 In Stock
10MG 188 In Stock
25MG 330 In Stock
50MG 479 In Stock
100MG 695 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    LSD1-IN-7 benzenesulfonate
  • Note
    Research use only, not for human use.
  • Brief Description
    LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
  • Description
    LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
  • In Vitro
    ——
  • In Vivo
    Animal Model:BALB/c nude mice bearing small cell lung carcinoma (SCLC)Dosage:5 mg/kg Administration:Oral administration; daily; for 30 days Result:Showed a tumor growth inhibition (TGI) of 78% at 5 mg/kg with nobody weight loss.
  • Synonyms
    CC-90011 benzenesulfonate
  • Pathway
    Chromatin/Epigenetic
  • Target
    Histone Demethylase
  • Recptor
    LSD1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2097523-60-7
  • Formula Weight
    609.64
  • Molecular Formula
    C30H29F2N5O5S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:60mg/ml(98.42mM; Need ultrasonic)
  • SMILES
    N#CC1=CC=C(C(N=C(N2CCC(N)CC2)N3C)=C(C4=CC=C(OC)C(F)=C4)C3=O)C=C1F.O=S(C5=CC=CC=C5)(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Young K. Chen, et al. Compositions comprising an inhibitor of lysine specific demethylase-1. WO2017079670A1.
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