Ticagrelor metabolite M5

CAS No. 1251765-07-7

Ticagrelor metabolite M5( AR-C133913XX | T437700 | Ticagrelor metabolite M5, )

Catalog No. M23421 CAS No. 1251765-07-7

Ticagrelor metabolite M5 is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 32 In Stock
5MG 55 In Stock
10MG 79 In Stock
25MG 159 In Stock
50MG 229 In Stock
100MG 310 In Stock
200MG 433 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Ticagrelor metabolite M5
  • Note
    Research use only, not for human use.
  • Brief Description
    Ticagrelor metabolite M5 is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor.
  • Description
    Ticagrelor metabolite M5 is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor. Compared to Clopidogrel, Ticagrelor has faster and more consistent inhibition on ADP-receptors. Ticagrelor is used in the treatment of acute coronary syndromes (ACS).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    AR-C133913XX | T437700 | Ticagrelor metabolite M5,
  • Pathway
    Neuroscience
  • Target
    P2 Receptor
  • Recptor
    P2Y12
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1251765-07-7
  • Formula Weight
    370.43
  • Molecular Formula
    C14H22N6O4S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:Soluble
  • SMILES
    CCCSC1=NC(=C2C(=N1)N(N=N2)[C@@H]3C[C@@H]([C@H]([C@H]3O)O)OCCO)N
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Teng R, Oliver S, Hayes MA, Butler K. Absorption, distribution, metabolism, and excretion of ticagrelor in healthy subjects. Drug Metab Dispos. 2010 Sep;38(9):1514-21. doi: 10.1124/dmd.110.032250. Epub 2010 Jun 15. PubMed PMID: 20551239.
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