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DMU2139
CAS No. 104890-70-2
DMU2139( —— )
Catalog No. M22628 CAS No. 104890-70-2
DMU2139 is a specific CYP1B1 inhibitor (CYP1B1 and CYP1A1 with IC50 of 9 nM and 795 nM, respectively).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 69 | In Stock |
|
| 5MG | 69 | In Stock |
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| 10MG | 112 | In Stock |
|
| 25MG | 226 | In Stock |
|
| 50MG | 327 | In Stock |
|
| 100MG | 486 | In Stock |
|
| 200MG | 704 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDMU2139
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NoteResearch use only, not for human use.
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Brief DescriptionDMU2139 is a specific CYP1B1 inhibitor (CYP1B1 and CYP1A1 with IC50 of 9 nM and 795 nM, respectively).
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DescriptionDMU2139 is a specific CYP1B1 inhibitor (CYP1B1 and CYP1A1 with IC50 of 9 nM and 795 nM, respectively).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetP450
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RecptorCYP1B1
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Research Area——
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Indication——
Chemical Information
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CAS Number104890-70-2
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Formula Weight289.3
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Molecular FormulaC19H15NO2
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Purity>98% (HPLC)
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Solubility——
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SMILESCOc1ccc2cc(ccc2c1)C(=O)\C=C\c1cccnc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Horley N J , Beresford K J M , Chawla T , et al. Discovery and characterization of novel CYP1B1 inhibitors based on heterocyclic chalcones: Overcoming cisplatin resistance in CYP1B1-overexpressing lines[J]. European Journal of Medicinal Chemistry, 2017, 129:159-174.
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