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CU-CPT-9a
CAS No. 2165340-32-7
CU-CPT-9a( —— )
Catalog No. M20662 CAS No. 2165340-32-7
CU-CPT-9a is a potent TLR8 inhibitor (IC50 : 0.5 nM) that suppresses TLR8-mediated proinflammatory signaling in various cell lines.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 85 | In Stock |
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| 2MG | 46 | In Stock |
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| 5MG | 76 | In Stock |
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| 10MG | 122 | In Stock |
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| 25MG | 237 | In Stock |
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| 50MG | 423 | In Stock |
|
| 100MG | 625 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCU-CPT-9a
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NoteResearch use only, not for human use.
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Brief DescriptionCU-CPT-9a is a potent TLR8 inhibitor (IC50 : 0.5 nM) that suppresses TLR8-mediated proinflammatory signaling in various cell lines.
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DescriptionCU-CPT-9a is a potent TLR8 inhibitor (IC50 : 0.5 nM) that suppresses TLR8-mediated proinflammatory signaling in various cell lines and human primary cells.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayImmunology/Inflammation
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TargetTLR
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RecptorTLR8
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Research Area——
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Indication——
Chemical Information
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CAS Number2165340-32-7
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Formula Weight265.31
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Molecular FormulaC17H15NO2
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Purity>98% (HPLC)
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SolubilityDMSO:150 mg/mL (565.38 mM)
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SMILESCOc1ccc2c(ccnc2c1)-c1ccc(O)c(C)c1
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Chemical Name2-Methyl-4-(7-methoxy-4-quinolinyl)phenol
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Zhang S Hu Z Tanji H et al. Small-molecule inhibition of TLR8 through stabilization of its resting state[J]. Nature Chemical Biology 2017 14(1):58-64.
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