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CPG-52364
CAS No. 1093135-60-4
CPG-52364( CPG 52364 | CPG52364 )
Catalog No. M10358 CAS No. 1093135-60-4
CPG-52364 (CPG52364) is an orally available, small molecule TLR7/8/9 antagonist for the treatment of systemic lupus erythematosus and other autoimmune disorders.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 376 | In Stock |
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| 10MG | 546 | In Stock |
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| 25MG | 842 | In Stock |
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| 50MG | 1107 | In Stock |
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| 100MG | 1516 | In Stock |
|
| 200MG | 2037 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCPG-52364
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NoteResearch use only, not for human use.
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Brief DescriptionCPG-52364 (CPG52364) is an orally available, small molecule TLR7/8/9 antagonist for the treatment of systemic lupus erythematosus and other autoimmune disorders.
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DescriptionCPG-52364 (CPG52364) is an orally available, small molecule TLR7/8/9 antagonist for the treatment of systemic lupus erythematosus and other autoimmune disorders.Other Indication Phase 1 Discontinued.
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In Vitro——
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In Vivo——
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SynonymsCPG 52364 | CPG52364
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PathwayImmunology/Inflammation
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TargetTLR
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RecptorTLR
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Research AreaOther Indications
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IndicationOther Disease
Chemical Information
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CAS Number1093135-60-4
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Formula Weight492.624
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Molecular FormulaC27H36N6O3
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Purity>98% (HPLC)
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Solubility——
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SMILESCN1CCN(C2=CC=C(C3=NC(NCCN4CCOCC4)=C5C=C(OC)C(OC)=CC5=N3)C=C2)CC1
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Chemical Name6,7-dimethoxy-2-(4-(4-methylpiperazin-1-yl)phenyl)-N-(2-morpholinoethyl)quinazolin-4-amine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Watanabe M, et al. ACS Med Chem Lett. 2014 Oct 2;5(11):1235-9.
2. Parkinson T. Curr Opin Mol Ther. 2008 Feb;10(1):21-31.
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