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LY2608204
CAS No. 1234703-40-2
LY2608204( LY-2608204 | LY 2608204 | LY2608204 )
Catalog No. M17209 CAS No. 1234703-40-2
LY2608204 has been used in trials studying the treatment of Diabetes Mellitus, Type 2.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 86 | In Stock |
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| 2MG | 43 | In Stock |
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| 5MG | 69 | In Stock |
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| 10MG | 93 | In Stock |
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| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLY2608204
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NoteResearch use only, not for human use.
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Brief DescriptionLY2608204 has been used in trials studying the treatment of Diabetes Mellitus, Type 2.
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DescriptionLY-2608204 is an activator of glucokinase (GK) with an EC50 value of 42 nM. LY2608204 decreases plasma glucose in a dose-dependent manner at both fasted and postprandial glucose levels. In 2010, LY-2608204 was entered clinical trials in Patients With Type 2 Diabetes.
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In Vitro——
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In Vivo——
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SynonymsLY-2608204 | LY 2608204 | LY2608204
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PathwayNeuroscience
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TargetGluR
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Recptorglucokinase
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Research AreaMetabolic Disease
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Indication——
Chemical Information
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CAS Number1234703-40-2
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Formula Weight559.81
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Molecular FormulaC28H37N3O3S3
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 100 mg/mL. 178.63 mM
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SMILESC1CCC(CC1)[C@@H]1C[C@]1(C(=O)Nc1ncc(s1)SCCN1CCCC1)c1ccc(cc1)S(=O)(=O)C1CC1
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Chemical Name(1R,2S)-2-cyclohexyl-1-(4-cyclopropylsulfonylphenyl)-N-[5-(2-pyrrolidin-1-ylethylsulfanyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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