CB-7921220

CAS No. 115453-99-1

CB-7921220( CB7921220 )

Catalog No. M10543 CAS No. 115453-99-1

CB-7921220 is a potent, selective Adenylyl Cyclase 1 (AC1) inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 35 Get Quote
5MG 78 Get Quote
10MG 132 Get Quote
25MG 285 Get Quote
50MG 483 Get Quote
100MG Get Quote Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    CB-7921220
  • Note
    Research use only, not for human use.
  • Brief Description
    CB-7921220 is a potent, selective Adenylyl Cyclase 1 (AC1) inhibitor.
  • Description
    CB-7921220 is a potent, selective Adenylyl Cyclase 1 (AC1) inhibitor.
  • In Vitro
    CB-7921220 shows a degree of isoform selectivity for adenylate cyclase (AC) 1, but cannot distinguish between AC1 and AC6. CB-7921220 has a more consistent predicted binding position in the two virtual docking screens, and has a binding conformation similar to ATP and P-site inhibitors, which may explain its lack of selectivity between AC1 and AC6.
  • In Vivo
    ——
  • Synonyms
    CB7921220
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Adenylate Cyclase
  • Recptor
    Adenylate Cyclase
  • Research Area
    Other Indications
  • Indication
    ——

Chemical Information

  • CAS Number
    115453-99-1
  • Formula Weight
    240.262
  • Molecular Formula
    C14H12N2O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : ≥ 100 mg/mL 416.22 mM
  • SMILES
    O=C(C1=NC(/C=C/C2=CC=C(N)C=C2)=CC=C1)O
  • Chemical Name
    6-[2-(4-aminophenyl)ethenyl]-2-pyridinecarboxylic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Brand CS, et al. J Pharmacol Exp Ther. 2013 Nov;347(2):265-75.
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