CB-7921220
CAS No. 115453-99-1
CB-7921220( CB7921220 )
Catalog No. M10543 CAS No. 115453-99-1
CB-7921220 is a potent, selective Adenylyl Cyclase 1 (AC1) inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 35 | Get Quote |
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| 5MG | 78 | Get Quote |
|
| 10MG | 132 | Get Quote |
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| 25MG | 285 | Get Quote |
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| 50MG | 483 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameCB-7921220
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NoteResearch use only, not for human use.
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Brief DescriptionCB-7921220 is a potent, selective Adenylyl Cyclase 1 (AC1) inhibitor.
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DescriptionCB-7921220 is a potent, selective Adenylyl Cyclase 1 (AC1) inhibitor.
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In VitroCB-7921220 shows a degree of isoform selectivity for adenylate cyclase (AC) 1, but cannot distinguish between AC1 and AC6. CB-7921220 has a more consistent predicted binding position in the two virtual docking screens, and has a binding conformation similar to ATP and P-site inhibitors, which may explain its lack of selectivity between AC1 and AC6.
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In Vivo——
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SynonymsCB7921220
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PathwayMetabolic Enzyme/Protease
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TargetAdenylate Cyclase
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RecptorAdenylate Cyclase
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Research AreaOther Indications
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Indication——
Chemical Information
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CAS Number115453-99-1
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Formula Weight240.262
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Molecular FormulaC14H12N2O2
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 100 mg/mL 416.22 mM
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SMILESO=C(C1=NC(/C=C/C2=CC=C(N)C=C2)=CC=C1)O
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Chemical Name6-[2-(4-aminophenyl)ethenyl]-2-pyridinecarboxylic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Brand CS, et al. J Pharmacol Exp Ther. 2013 Nov;347(2):265-75.
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