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CK2α-IN-1
CAS No. 443747-52-2
CK2α-IN-1( —— )
Catalog No. M36508 CAS No. 443747-52-2
CK2α-IN-1 is a selective non-ATP-competitive CK2α inhibitor with an IC50 of 7.0 μM and a Ki of 1.6 μM.CK2α-IN-1 exhibits potential anticancer activity and can be used in cancer research.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 55 | Get Quote |
|
| 5MG | 77 | Get Quote |
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| 10MG | 113 | Get Quote |
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| 25MG | 200 | Get Quote |
|
| 50MG | 339 | Get Quote |
|
| 100MG | 611 | Get Quote |
|
| 500MG | 1287 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameCK2α-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionCK2α-IN-1 is a selective non-ATP-competitive CK2α inhibitor with an IC50 of 7.0 μM and a Ki of 1.6 μM.CK2α-IN-1 exhibits potential anticancer activity and can be used in cancer research.
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DescriptionCK2α-IN-1 (compound 2) is a selective CK2α inhibitor (IC50=7.0 μM; Ki=1.6 μM) that exhibits a non-ATP-competitive mode of action. CK2α-IN-1 exhibits good potential for anticancer studies.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetCasein Kinase
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RecptorCasein Kinase
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Research Area——
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Indication——
Chemical Information
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CAS Number443747-52-2
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Formula Weight341.34
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Molecular FormulaC16H11N3O4S
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Purity>98% (HPLC)
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Solubility——
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SMILESN(C1=NC(=CS1)C2=CC(N(=O)=O)=CC=C2)C3=CC(C(O)=O)=CC=C3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Bestgen B, et al. 2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 1. Identification of an Allosteric Binding Site. J Med Chem. 2019 Feb 28;62(4):1803-1816. ?
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