Rapastinel( GLYX-13 | Thr-Pro-Pro-Thr-NH2 )

Catalog No. M10606 CAS No. 117928-94-6

A tetrapeptide (TPPT-amide) that acts as a NMDA receptor glycine site partial agonist.

Purity : >98% (HPLC)

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HNMR

HPLC

MSDS

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Biological Information

Product Name

Rapastinel
Note

Research use only, not for human use.
Brief Description

A tetrapeptide (TPPT-amide) that acts as a NMDA receptor glycine site partial agonist.
Description

A tetrapeptide (TPPT-amide) that acts as a NMDA receptor glycine site partial agonist; readily crosses the blood-brain barrier and modulates the NMDA receptor, shows potent cognitive-enhancing properties in a valid in vivo model of learning.Depression Phase 3 Clinical.
In Vitro

——
In Vivo

——
Synonyms

GLYX-13 | Thr-Pro-Pro-Thr-NH2
Pathway

Membrane Transporter/Ion Channel
Target

iGluR
Recptor

Others
Research Area

Neurological Disease
Indication

Depression

Chemical Information

CAS Number

117928-94-6
Formula Weight

413.4686
Molecular Formula

C18H31N5O6
Purity

>98% (HPLC)
Solubility

DMSO: ≥ 32 mg/mL
SMILES

C[C@@H](O)[C@@H](C(N)=O)NC([C@H]1N(C([C@H]2N(C([C@H]([C@H](O)C)N)=O)CCC2)=O)CCC1)=O
Chemical Name

L-Threoninamide, L-threonyl-L-prolyl-L-prolyl-

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Moskal JR, et al. Neuropharmacology. 2005 Dec;49(7):1077-87. 2. Zhang XL, et al. Neuropharmacology. 2008 Dec;55(7):1238-50. 3. Burgdorf J, et al. Neurobiol Aging. 2011 Apr;32(4):698-706.

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