Nefopam hydrochloride

CAS No. 23327-57-3

Nefopam hydrochloride( —— )

Catalog No. M13669 CAS No. 23327-57-3

Nefopam hydrochloride is a centrally-acting but non-opioid analgesic drug by blocking voltage-gated sodium channel and inhibition of serotonin, dopamine and noradrenaline reuptake.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
10MG 32 In Stock
25MG 41 In Stock
50MG 59 In Stock
100MG 106 In Stock
200MG 178 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Nefopam hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Nefopam hydrochloride is a centrally-acting but non-opioid analgesic drug by blocking voltage-gated sodium channel and inhibition of serotonin, dopamine and noradrenaline reuptake.
  • Description
    Nefopam hydrochloride is a centrally-acting but non-opioid analgesic drug by blocking voltage-gated sodium channel and inhibition of serotonin, dopamine and noradrenaline reuptake.(In Vitro):Nefopam hydrochloride (Fenazoxine hydrochloride) is a non-opioid, non-steroidal, centrally acting analgesic drug that is derivative of the non-sedative benzoxazocine. Constitutively elevated β-catenin leads to a delayed and fibrous fracture repair process, and Nefopam inhibits β-catenin mediated signaling during skin wound repair.
  • In Vitro
    Nefopam hydrochloride (Fenazoxine hydrochloride) is a non-opioid, non-steroidal, centrally acting analgesic drug that is derivative of the non-sedative benzoxazocine.Constitutively elevated β-catenin leads to a delayed and fibrous fracture repair process, and Nefopam inhibits β-catenin mediated signaling during skin wound repair.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    Sodium Channel
  • Recptor
    Sodium Channel
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    23327-57-3
  • Formula Weight
    289.8
  • Molecular Formula
    C17H20ClNO
  • Purity
    >98% (HPLC)
  • Solubility
    Water: 21 mg/mL (72.46 mM); DMSO: 1 mg/mL (3.45 mM)
  • SMILES
    Cl.CN1CCOC(C2=CC=CC=C2)C2=CC=CC=C2C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. M. S. Evans1, et al, lBr J Anaesth, 2008, 101(5), 610-617.
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