Vepafestinib

CAS No. 2129515-96-2

Vepafestinib( —— )

Catalog No. M37628 CAS No. 2129515-96-2

Vepafestinib is a RET inhibitor with potential antineoplastic activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Vepafestinib
  • Note
    Research use only, not for human use.
  • Brief Description
    Vepafestinib is a RET inhibitor with potential antineoplastic activity.
  • Description
    Vepafestinib (TAS0953/HM06; compound 6) is a RET inhibitor (extracted from patent WO2019039439). Vepafestinib is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Tyrosine Kinase
  • Target
    c-RET
  • Recptor
    c-RET
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2129515-96-2
  • Formula Weight
    474.55
  • Molecular Formula
    C26H30N6O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 50 mg/mL (105.36 mM; Ultrasonic )
  • SMILES
    COCc1ccc(NC(=O)c2c(C#CCN3CCOCC3)n(c3ncnc(N)c23)C2(C)CC2)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Hayashi, Kohei, et al. FUSION PROTEIN OF DCTN1 PROTEIN WITH RET PROTEIN. WO2019039439.
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