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DUN73423
CAS No. 2414373-42-3
DUN73423( —— )
Catalog No. M36296 CAS No. 2414373-42-3
DUN73423 (RET-IN-21) is a potent tyrosine kinase (RET) inhibitor with antitumour activity for the study of cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 73 | Get Quote |
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| 5MG | 117 | Get Quote |
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| 10MG | 180 | Get Quote |
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| 25MG | 296 | Get Quote |
|
| 50MG | 441 | Get Quote |
|
| 100MG | 618 | Get Quote |
|
| 500MG | 1251 | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameDUN73423
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NoteResearch use only, not for human use.
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Brief DescriptionDUN73423 (RET-IN-21) is a potent tyrosine kinase (RET) inhibitor with antitumour activity for the study of cancer.
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DescriptionRET-IN-21 is an inhibitor of receptor tyrosine kinase (RET), with the IC50 of 4.4 μM, that has antitumor activity.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayTyrosine Kinase
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Targetc-RET
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Recptorc-RET
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Research Area——
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Indication——
Chemical Information
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CAS Number2414373-42-3
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Formula Weight344.37
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Molecular FormulaC19H16N6O
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Purity>98% (HPLC)
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Solubility——
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SMILESN(CC=1C=CN=CC1)C2=NC3=C(C=NN3C=C2)C4=CC=C(C(N)=O)C=C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Rebecca Newton, et al. Discovery and Optimization of wt-RET/KDR-Selective Inhibitors of RETV804M Kinase. ACS Med. Chem. Lett. 2020, 11, 4, 497–505
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