Opevesostat

CAS No. 2231294-96-3

Opevesostat( —— )

Catalog No. M37000 CAS No. 2231294-96-3

Opevesostat (ODM-208) is an inhibitor of lyase (CYP11A1) (the enzyme cleavage cholesterol side chain).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 67 In Stock
5MG 61 In Stock
10MG 101 In Stock
25MG 188 In Stock
50MG 291 In Stock
100MG 431 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Opevesostat
  • Note
    Research use only, not for human use.
  • Brief Description
    Opevesostat (ODM-208) is an inhibitor of lyase (CYP11A1) (the enzyme cleavage cholesterol side chain).
  • Description
    Opevesostat is a cholesterol side-chain cleavage enzyme (CYP11A1) inhibitor.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    P450
  • Recptor
    P450
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2231294-96-3
  • Formula Weight
    418.51
  • Molecular Formula
    C21H26N2O5S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 50 mg/mL (119.47 mM; Ultrasonic )
  • SMILES
    C(N1CC=2C(C1)=CC=CC2)C3=CC(=O)C(OCC4CCN(S(C)(=O)=O)CC4)=CO3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ikonen, et al. Method for treating prostate cancer in patient using CYP11A1 inhibitor as active ingredient. World Intellectual Property Organization, WO2023052682 A1. 2023-04-06.
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