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Opevesostat
CAS No. 2231294-96-3
Opevesostat( —— )
Catalog No. M37000 CAS No. 2231294-96-3
Opevesostat (ODM-208) is an inhibitor of lyase (CYP11A1) (the enzyme cleavage cholesterol side chain).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 67 | In Stock |
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| 5MG | 61 | In Stock |
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| 10MG | 101 | In Stock |
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| 25MG | 188 | In Stock |
|
| 50MG | 291 | In Stock |
|
| 100MG | 431 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameOpevesostat
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NoteResearch use only, not for human use.
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Brief DescriptionOpevesostat (ODM-208) is an inhibitor of lyase (CYP11A1) (the enzyme cleavage cholesterol side chain).
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DescriptionOpevesostat is a cholesterol side-chain cleavage enzyme (CYP11A1) inhibitor.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetP450
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RecptorP450
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Research Area——
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Indication——
Chemical Information
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CAS Number2231294-96-3
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Formula Weight418.51
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Molecular FormulaC21H26N2O5S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (119.47 mM; Ultrasonic )
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SMILESC(N1CC=2C(C1)=CC=CC2)C3=CC(=O)C(OCC4CCN(S(C)(=O)=O)CC4)=CO3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ikonen, et al. Method for treating prostate cancer in patient using CYP11A1 inhibitor as active ingredient. World Intellectual Property Organization, WO2023052682 A1. 2023-04-06.
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