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PERK-IN-6
CAS No. 1337532-14-5
PERK-IN-6( —— )
Catalog No. M36418 CAS No. 1337532-14-5
PERK-IN-6 is a novel and highly potent PERK inhibitor (IC50:2.5 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 375 | In Stock |
|
| 10MG | 559 | In Stock |
|
| 25MG | 892 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePERK-IN-6
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NoteResearch use only, not for human use.
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Brief DescriptionPERK-IN-6 is a novel and highly potent PERK inhibitor (IC50:2.5 nM).
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DescriptionPERK-IN-6 (Compound 5) is a PERK inhibitor with an IC50 of 2.5 nM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayApoptosis
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TargetPERK
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RecptorPERK
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Research Area——
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Indication——
Chemical Information
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CAS Number1337532-14-5
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Formula Weight398.46
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Molecular FormulaC23H22N6O
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Purity>98% (HPLC)
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Solubility——
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SMILESNC1=C2C(=CN(C)C2=NC=N1)C=3C=C4C(=CC3)N(C(CC=5N=C(C)C=CC5)=O)CC4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Axten JM, et al. Discovery of GSK2656157: An Optimized PERK Inhibitor Selected for Preclinical Development. ACS Med Chem Lett. 2013 Aug 12;4(10):964-8.?
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