PERK-IN-6

CAS No. 1337532-14-5

PERK-IN-6( —— )

Catalog No. M36418 CAS No. 1337532-14-5

PERK-IN-6 is a novel and highly potent PERK inhibitor (IC50:2.5 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 375 In Stock
10MG 559 In Stock
25MG 892 In Stock
100MG Get Quote In Stock
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Biological Information

  • Product Name
    PERK-IN-6
  • Note
    Research use only, not for human use.
  • Brief Description
    PERK-IN-6 is a novel and highly potent PERK inhibitor (IC50:2.5 nM).
  • Description
    PERK-IN-6 (Compound 5) is a PERK inhibitor with an IC50 of 2.5 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Apoptosis
  • Target
    PERK
  • Recptor
    PERK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1337532-14-5
  • Formula Weight
    398.46
  • Molecular Formula
    C23H22N6O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    NC1=C2C(=CN(C)C2=NC=N1)C=3C=C4C(=CC3)N(C(CC=5N=C(C)C=CC5)=O)CC4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Axten JM, et al. Discovery of GSK2656157: An Optimized PERK Inhibitor Selected for Preclinical Development. ACS Med Chem Lett. 2013 Aug 12;4(10):964-8.?
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