Cart
sales@molnova.com
p53-MDM2-IN-1
CAS No. 381717-91-5
p53-MDM2-IN-1( —— )
Catalog No. M36397 CAS No. 381717-91-5
p53-MDM2-IN-1 (Example 30), an inhibitor of the p53-MDM2/X protein interaction, exhibits a K i value of 23.35 μM and holds potential for applications in anti-tumor research.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 278 | In Stock |
|
| 10MG | 408 | In Stock |
|
| 25MG | 620 | In Stock |
|
| 50MG | 826 | In Stock |
|
| 100MG | 1097 | In Stock |
|
| 200MG | 1469 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product Namep53-MDM2-IN-1
-
NoteResearch use only, not for human use.
-
Brief Descriptionp53-MDM2-IN-1 (Example 30), an inhibitor of the p53-MDM2/X protein interaction, exhibits a K i value of 23.35 μM and holds potential for applications in anti-tumor research.
-
Descriptionp53-MDM2-IN-1 (Example 30) is an inhibitor of p53-MDM2/X protein interaction with an Ki value of 23.35 μM. p53-MDM2-IN-1 can be used for anti-tumor research.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayApoptosis
-
TargetMDM2-p53
-
RecptorMdm2 | p53
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number381717-91-5
-
Formula Weight421.88
-
Molecular FormulaC23H20ClN3O3
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESC(=O)(C=1C(N(CCCN2C=CN=C2)C(=O)C1O)C3=CC=C(Cl)C=C3)C4=CC=CC=C4
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Zhang W, et al. Pyrrylketone compound and application thereof as drug. China. CN102603717.
molnova catalog
related products
-
UNC-2170
UNC-2170 is a small molecule ligand for the methyl-lysine binding protein 53BP1 (p53-binding protein 1) with Kd of 22 uM against the 53BP1 tandem tudor domain.
-
MI 219
MI 219 is a potent, specific MDM2-p53 inhibitor with Ki of 5 nM, >10,000-fold selective for MDM2 over MDMX.
-
Pifithrin-β hydrobro...
A cyclic analog of Pifithrin-α and a small molecule inhibitor of p53; prevents dexamethasone-induced cell death in murine thymocytes with EC50 of 2.01 uM.
