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PF-07258669
CAS No. 2755890-53-8
PF-07258669( —— )
Catalog No. M36282 CAS No. 2755890-53-8
PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 1284 | Get Quote |
|
| 5MG | 1606 | Get Quote |
|
| 10MG | 2613 | Get Quote |
|
| 25MG | 4996 | Get Quote |
|
| 50MG | 7995 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePF-07258669
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NoteResearch use only, not for human use.
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Brief DescriptionPF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.
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DescriptionPF-07258669 is a melanocortin-4 receptor (MC4) antagonist. PF-07258669 can be used for the research of cachexia, anorexia, or anorexia nervosa.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetMelanocortin Receptor
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RecptorMelanocortin Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2755890-53-8
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Formula Weight462.52
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Molecular FormulaC25H27FN6O2
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Purity>98% (HPLC)
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Solubility——
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SMILESC([C@H](C)C=1C=C(OC)N=CC1F)(=O)N2C[C@@]3(NC=4C(CC3)=CC(=C(C)N4)C=5N=CC=CN5)CC2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Christopher Ryan BUTLER, et al. Spiro compounds as melanocortin 4 receptor antagonists and uses thereof. Patent. WO2021250541A1.
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