Cart
sales@molnova.com
Dual FAAH/sEH-IN-1
CAS No. 2756099-59-7
Dual FAAH/sEH-IN-1( —— )
Catalog No. M35726 CAS No. 2756099-59-7
Dual FAAH/sEH-IN-1 is a dual inhibitor of sEH (soluble epoxide hydrolase) (IC50: 9.6 nM) and FAAH (fatty acid amide hydrolase) (IC50: 7 nM) with high affinity and anti-inflammatory activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 285 | In Stock |
|
| 5MG | 231 | In Stock |
|
| 10MG | 307 | In Stock |
|
| 25MG | 466 | In Stock |
|
| 50MG | 613 | In Stock |
|
| 100MG | 820 | In Stock |
|
| 200MG | 1088 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameDual FAAH/sEH-IN-1
-
NoteResearch use only, not for human use.
-
Brief DescriptionDual FAAH/sEH-IN-1 is a dual inhibitor of sEH (soluble epoxide hydrolase) (IC50: 9.6 nM) and FAAH (fatty acid amide hydrolase) (IC50: 7 nM) with high affinity and anti-inflammatory activity.
-
DescriptionDual FAAH/sEH-IN-1 (compound 3) is a high affinity dual sEH (soluble epoxide hydrolase) and FAAH (fatty acid amide hydrolase) inhibitor, with IC50 values of 9.6 and 7 nM, respectively. Dual FAAH/sEH-IN-1 shows antinociception against the inflammatory phase.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayMetabolic Enzyme/Protease
-
TargetFAAH
-
RecptorFAAH | Epoxide Hydrolase
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2756099-59-7
-
Formula Weight512.04
-
Molecular FormulaC25H22ClN3O3S2
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESN(C(=O)C1CCN(S(=O)(=O)C2=C(Cl)C=CC=C2)CC1)C3=CC=C(C4=NC=5C(S4)=CC=CC5)C=C3
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Wilt S, Kodani S, Valencia L, et al. Further exploration of the structure-activity relationship of dual soluble epoxide hydrolase/fatty acid amide hydrolase inhibitors. Bioorg Med Chem. 2021;51:116507.?
molnova catalog
related products
-
PDM2
PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.
-
PF-3845
PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.
-
MM-433593
MM-433593 is a selective fatty acid amide hydrolase (FAAH-1) inhibitor for the treatment of pain, inflammation, and other disorders.
