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Home - Products - Metabolic Enzyme/Protease - FAAH - PDM2

PDM2

CAS No. 688348-25-6

PDM2( —— )

Catalog No. M18999 CAS No. 688348-25-6

PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    PDM2
  • Note
    Research use only, not for human use.
  • Brief Description
    PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.
  • Description
    PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.
  • In Vitro
    PDM2 (Compound 4b) exhibits a Ki of 1.2±0.4 nM for AhR and no affinity for estrogen receptor (ER), confirming that replacement of hydroxyl with chloride abolished binding on ER and increased dramatically the affinity for AhR.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    FAAH
  • Recptor
    AhR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    688348-25-6
  • Formula Weight
    283.58
  • Molecular Formula
    C14H9Cl3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : 50 mg/mL 176.32 mM
  • SMILES
    Clc1ccc(cc1)\C=C\c1cc(Cl)cc(Cl)c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.de Medina, P. ,Casper, R.,Savouret, J.F., et al. Journal of Medicinal Chemistry 48, 287-291 (2005).
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