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DS12881479
CAS No. 2373065-59-7
DS12881479( —— )
Catalog No. M35456 CAS No. 2373065-59-7
DS12881479 can be used in cancer research which is a potent and selective inhibitor of Mnk1(IC 50 =21 nM) .
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 244 | In Stock |
|
| 10MG | 368 | In Stock |
|
| 25MG | 661 | In Stock |
|
| 50MG | 870 | In Stock |
|
| 100MG | 1144 | In Stock |
|
| 200MG | 1562 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDS12881479
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NoteResearch use only, not for human use.
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Brief DescriptionDS12881479 can be used in cancer research which is a potent and selective inhibitor of Mnk1(IC 50 =21 nM) .
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DescriptionDS12881479 is a potent and selective Mnk1 inhibitor with an IC50 value of 21 nM. DS12881479 can be used in cancer research.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMAPK/ERK Signaling
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TargetMNK
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RecptorMNK
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Research Area——
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Indication——
Chemical Information
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CAS Number2373065-59-7
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Formula Weight301.41
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Molecular FormulaC16H19N3OS
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (829.43 mM; Ultrasonic )
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SMILESCN1CCC(CC1)C(=O)Nc1ncc(s1)-c1ccccc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Yumi Matsui, et al. A novel inhibitor stabilizes the inactive conformation of MAPK-interacting kinase 1. Acta Crystallogr F Struct Biol Commun. 2018 Mar 1;74(Pt 3):156-160.?
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