MNK1/2-IN-5

CAS No. 1426928-20-2

MNK1/2-IN-5( —— )

Catalog No. M35464 CAS No. 1426928-20-2

MNK1/2-IN-5 is a potent and selective MNK1/2 inhibitor with anticancer activity and can be used to study solid tumors and hematological malignancies.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 141 In Stock
2MG 79 In Stock
5MG 132 In Stock
10MG 198 In Stock
25MG 356 In Stock
50MG 513 In Stock
100MG 732 In Stock
200MG 1004 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    MNK1/2-IN-5
  • Note
    Research use only, not for human use.
  • Brief Description
    MNK1/2-IN-5 is a potent and selective MNK1/2 inhibitor with anticancer activity and can be used to study solid tumors and hematological malignancies.
  • Description
    MNK1/2-IN-5 is a potent and selective MNK1/2 inhibitor as a therapeutic agent.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    MAPK/ERK Signaling
  • Target
    MNK
  • Recptor
    MNK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1426928-20-2
  • Formula Weight
    308.33
  • Molecular Formula
    C17H16N4O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 7.14 mg/mL (23.16 mM; Ultrasonic (<60°C)
  • SMILES
    O([C@@H](CN)C)C1=NN2C(=CN=C2C=C1)C3=CC=4C(O3)=CC=CC4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Xu W, et al. Update on the Development of MNK Inhibitors as Therapeutic Agents. J Med Chem. 2021 Sep 17.?
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