MNK1/2-IN-5

CAS No. 1426928-20-2

MNK1/2-IN-5( —— )

Catalog No. M35464 CAS No. 1426928-20-2

MNK1/2-IN-5 is a potent and selective MNK1/2 inhibitor with anticancer activity and can be used to study solid tumors and hematological malignancies.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 88 Get Quote
5MG 132 Get Quote
10MG 211 Get Quote
25MG 345 Get Quote
50MG 508 Get Quote
100MG 708 Get Quote
500MG 1431 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    MNK1/2-IN-5
  • Note
    Research use only, not for human use.
  • Brief Description
    MNK1/2-IN-5 is a potent and selective MNK1/2 inhibitor with anticancer activity and can be used to study solid tumors and hematological malignancies.
  • Description
    MNK1/2-IN-5 is a potent and selective MNK1/2 inhibitor as a therapeutic agent.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    MAPK/ERK Signaling
  • Target
    MNK
  • Recptor
    MNK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1426928-20-2
  • Formula Weight
    308.33
  • Molecular Formula
    C17H16N4O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 7.14 mg/mL (23.16 mM; Ultrasonic (<60°C)
  • SMILES
    O([C@@H](CN)C)C1=NN2C(=CN=C2C=C1)C3=CC=4C(O3)=CC=CC4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Xu W, et al. Update on the Development of MNK Inhibitors as Therapeutic Agents. J Med Chem. 2021 Sep 17.?
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