YAP/TAZ inhibitor-2?

CAS No. 2762617-31-0

YAP/TAZ inhibitor-2?( —— )

Catalog No. M35381 CAS No. 2762617-31-0

YAP/TAZ inhibitor-2 is a potent, orally active TEAD-YAP/TAZ inhibitor with an EC50 value of 3 nM, demonstrating anti-proliferative and antitumor activity .

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 128 Get Quote
5MG 187 Get Quote
10MG 297 Get Quote
25MG 486 Get Quote
50MG 702 Get Quote
100MG 963 Get Quote
500MG 1917 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    YAP/TAZ inhibitor-2?
  • Note
    Research use only, not for human use.
  • Brief Description
    YAP/TAZ inhibitor-2 is a potent, orally active TEAD-YAP/TAZ inhibitor with an EC50 value of 3 nM, demonstrating anti-proliferative and antitumor activity .
  • Description
    YAP/TAZ inhibitor-2 is a potent and orally active TEAD-YAP/TAZ inhibitor with an EC50 value of 3 nM. YAP/TAZ inhibitor-2 shows anti-proliferative activity. YAP/TAZ inhibitor-2 shows antitumor activity.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    YAP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2762617-31-0
  • Formula Weight
    390.33
  • Molecular Formula
    C19H14F4N4O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (256.19 mM; Ultrasonic )
  • SMILES
    FC(=C)C(=O)N1CC(C1)n1nc(-c2ccc(cc2)C(F)(F)F)c2cccnc12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Xu, xiaofeng, et al. Bicyclic compounds, compositions and use thereof. WO2022037568A1.
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