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CAY10462
CAS No. 502656-68-0
CAY10462( —— )
Catalog No. M34986 CAS No. 502656-68-0
CAY10462 (CTK8E8405) is an effective and selective inhibitor of the 20-HETE synthase CYP4A11 with an IC50 of 8.8 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 28 | In Stock |
|
| 5MG | 46 | In Stock |
|
| 10MG | 84 | In Stock |
|
| 25MG | 204 | In Stock |
|
| 50MG | 300 | In Stock |
|
| 100MG | 433 | In Stock |
|
| 200MG | 603 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCAY10462
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NoteResearch use only, not for human use.
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Brief DescriptionCAY10462 (CTK8E8405) is an effective and selective inhibitor of the 20-HETE synthase CYP4A11 with an IC50 of 8.8 nM.
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DescriptionCAY 10434 dihydrochloride is a potent CYP4A hydroxylase inhibitor. CAY 10434 dihydrochloride improves contractile response to angiotensin II with the maximal contractile response (Emax) 6764 mg.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetP450
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RecptorP450
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Research Area——
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Indication——
Chemical Information
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CAS Number502656-68-0
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Formula Weight360.32
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Molecular FormulaC17H27Cl2N3O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 35.71 mg/mL (99.11 mM; Ultrasonic (<60°C)
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SMILESCN(C)CCCCCCOC(C=C1)=CC=C1N2C=CN=C2.Cl.Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Jerez S, et al. 17-Octadecynoic acid improves contractile response to angiotensin II by releasing vasocontrictor prostaglandins. Prostaglandins Other Lipid Mediat. 2012 Jan;97(1-2):36-42. ?
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