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Aplindore Fumarate

CAS No. 189681-71-8

Aplindore Fumarate( —— )

Catalog No. M34505 CAS No. 189681-71-8

Aplindore Fumarate (DAB-452) is a small molecule dopamine D2 receptor partial agonist.Aplindore Fumarate exhibits high affinity for dopamine D2 and D3 receptors, and low affinity for dopamine D4, 5-hydroxytryptophan (5-HT2), and α1-adrenergic receptors.

Purity : >98% (HPLC)

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Size	Price / USD	Stock	Quantity
2MG	445	Get Quote
5MG	696	Get Quote
10MG	938	Get Quote
25MG	1408	Get Quote
50MG	1822	Get Quote
100MG	2520	Get Quote
500MG	Get Quote	Get Quote
1G	Get Quote	Get Quote

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Biological Information

Product Name

Aplindore Fumarate
Note

Research use only, not for human use.
Brief Description

Aplindore Fumarate (DAB-452) is a small molecule dopamine D2 receptor partial agonist.Aplindore Fumarate exhibits high affinity for dopamine D2 and D3 receptors, and low affinity for dopamine D4, 5-hydroxytryptophan (5-HT2), and α1-adrenergic receptors.
Description

Aplindore Fumarate (DAB-452) is a small molecule dopamine D2 receptor partial agonist.Aplindore Fumarate exhibits high affinity for dopamine D2 and D3 receptors, and low affinity for dopamine D4, 5-hydroxytryptophan (5-HT2), and α1-adrenergic receptors.Aplindore Fumarate is used in the study of Parkinson's disease and schizophrenia. Fumarate can be used to study Parkinson's and schizophrenia.
In Vitro

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In Vivo

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Synonyms

——
Pathway

GPCR/G Protein
Target

Dopamine Receptor
Recptor

Dopamine Receptor | 5-HT Receptor | Adrenergic Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

189681-71-8
Formula Weight

426.42
Molecular Formula

C22H22N2O7
Purity

>98% (HPLC)
Solubility

——
SMILES

C(=C/C(O)=O)\C(O)=O.C(NCC1=CC=CC=C1)[C@@H]2OC=3C4=C(C=CC3OC2)NC(=O)C4
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

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