IK-862

CAS No. 478911-60-3

IK-862( —— )

Catalog No. M34281 CAS No. 478911-60-3

IK-862 is a selective inhibitor of TACE (ADAM17).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 848 In Stock
10MG 1159 In Stock
25MG 1701 In Stock
50MG 2279 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    IK-862
  • Note
    Research use only, not for human use.
  • Brief Description
    IK-862 is a selective inhibitor of TACE (ADAM17).
  • Description
    IK-862 is a selective inhibitor of TACE.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    MMP
  • Recptor
    MMP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    478911-60-3
  • Formula Weight
    433.5
  • Molecular Formula
    C25H27N3O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C[C@@]1(C(=O)N([C@@H](C(NO)=O)C)CC1)C2=CC=C(OCC=3C4=C(N=C(C)C3)C=CC=C4)C=C2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Georgiadis D, et al. Specific targeting of metzincin family members with small-molecule inhibitors: progress toward a multifarious challenge. Bioorg Med Chem. 2008;16(19):8781-8794. doi:10.1016/j.bmc.2008.08.058?
molnova catalog
related products
  • Marimastat

    A broad spectrum MMP inhibitor for MMP9/1/2/14/7 with IC50 of 3/5/6/9/13 nM, respectively.

  • SB-3CT

    SB-3CT is an effective and selective gelatinase inhibitor with Ki of 13.9 nM and 600 nM for MMP-2 and MMP-9, respectively.

  • MMP2-IN-3

    MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM). MMP2-IN-3 inhibits MMP-9 and MMP-8 with IC50s of 26.6 and 32 μM, respectively.