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GPR35 agonist 2
CAS No. 494191-73-0
GPR35 agonist 2( —— )
Catalog No. M33937 CAS No. 494191-73-0
GPR35 agonist 2 (TC-G 1001) is a potent GPR35 agonist.The EC50 values of GPR35 agonist 2 in the β-arrestin and Ca2+ release assays were 26 and 3.2 nM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 110 | In Stock |
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| 5MG | 92 | In Stock |
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| 10MG | 169 | In Stock |
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| 25MG | 377 | In Stock |
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| 50MG | 548 | In Stock |
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| 100MG | 784 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 1609 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGPR35 agonist 2
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NoteResearch use only, not for human use.
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Brief DescriptionGPR35 agonist 2 (TC-G 1001) is a potent GPR35 agonist.The EC50 values of GPR35 agonist 2 in the β-arrestin and Ca2+ release assays were 26 and 3.2 nM, respectively.
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DescriptionGPR35 agonist 2 (compound 11) is a potent agonist of GPR35, with EC50s of 26 and 3.2 nM in the β-arrestin and Ca2+ release assay, respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetGPR
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RecptorGPR
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Research Area——
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Indication——
Chemical Information
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CAS Number494191-73-0
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Formula Weight342.34
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Molecular FormulaC17H11FN2O3S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 25 mg/mL (73.03 mM; Ultrasonic )
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SMILESOC(=O)c1ccc(\C=C2\SC(Nc3ccccc3F)=NC2=O)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Thimm D, et, al. 6-Bromo-8-(4-[(3)H]methoxybenzamido)-4-oxo-4H-chromene-2-carboxylic Acid: a powerful tool for studying orphan G protein-coupled receptor GPR35. J Med Chem. 2013 Sep 12; 56(17): 7084-99.?
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