CBiPES hydrochloride

CAS No. 856702-40-4

CBiPES hydrochloride( —— )

Catalog No. M33836 CAS No. 856702-40-4

CBiPES hydrochloride (CBiPES HCl) is a potent orthosteric modulator of the mGlu2 receptor with an EC50 value of 92.8 nM.CBiPES hydrochloride blocks the action of WT and mGlu(3) receptors.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 263 Get Quote
5MG 416 Get Quote
10MG 603 Get Quote
25MG 906 Get Quote
50MG 1214 Get Quote
100MG 1611 Get Quote
500MG 3231 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    CBiPES hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    CBiPES hydrochloride (CBiPES HCl) is a potent orthosteric modulator of the mGlu2 receptor with an EC50 value of 92.8 nM.CBiPES hydrochloride blocks the action of WT and mGlu(3) receptors.
  • Description
    CBiPES hydrochloride is a mGlu2 receptor positive allosteric modulator (EC50: 92.8 nM). CBiPES hydrochloride attenuates stress-induced hyperthermia and PCP-induced hyperlocomotor activity. CBiPES hydrochloride can be used for research of neurological disease.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Neuroscience
  • Target
    GluR
  • Recptor
    GluR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    856702-40-4
  • Formula Weight
    413.92
  • Molecular Formula
    C21H20ClN3O2S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cl.N#CC1=CC=C(C=C1)C=2C=CC=C(C2)N(CC=3C=NC=CC3)S(=O)(=O)CC
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Johnson MP, et al. Metabotropic glutamate 2 receptor potentiators: receptor modulation, frequency-dependent synaptic activity, and efficacy in preclinical anxiety and psychosis model(s). Psychopharmacology (Berl). 2005 Apr;179(1):271-83.?
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