CBiPES hydrochloride
CAS No. 856702-40-4
CBiPES hydrochloride( —— )
Catalog No. M33836 CAS No. 856702-40-4
CBiPES hydrochloride (CBiPES HCl) is a potent orthosteric modulator of the mGlu2 receptor with an EC50 value of 92.8 nM.CBiPES hydrochloride blocks the action of WT and mGlu(3) receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 263 | Get Quote |
|
| 5MG | 416 | Get Quote |
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| 10MG | 603 | Get Quote |
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| 25MG | 906 | Get Quote |
|
| 50MG | 1214 | Get Quote |
|
| 100MG | 1611 | Get Quote |
|
| 500MG | 3231 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameCBiPES hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionCBiPES hydrochloride (CBiPES HCl) is a potent orthosteric modulator of the mGlu2 receptor with an EC50 value of 92.8 nM.CBiPES hydrochloride blocks the action of WT and mGlu(3) receptors.
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DescriptionCBiPES hydrochloride is a mGlu2 receptor positive allosteric modulator (EC50: 92.8 nM). CBiPES hydrochloride attenuates stress-induced hyperthermia and PCP-induced hyperlocomotor activity. CBiPES hydrochloride can be used for research of neurological disease.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayNeuroscience
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TargetGluR
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RecptorGluR
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Research Area——
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Indication——
Chemical Information
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CAS Number856702-40-4
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Formula Weight413.92
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Molecular FormulaC21H20ClN3O2S
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Purity>98% (HPLC)
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Solubility——
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SMILESCl.N#CC1=CC=C(C=C1)C=2C=CC=C(C2)N(CC=3C=NC=CC3)S(=O)(=O)CC
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Johnson MP, et al. Metabotropic glutamate 2 receptor potentiators: receptor modulation, frequency-dependent synaptic activity, and efficacy in preclinical anxiety and psychosis model(s). Psychopharmacology (Berl). 2005 Apr;179(1):271-83.?
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