Fluorobexarotene( —— )

Catalog No. M32926 CAS No. 1190848-23-7

Fluorobexarotene possesses an apparent RXR binding affinity that is 75% greater than Bexarotene.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	354	In Stock
5MG	440	In Stock
10MG	649	In Stock
25MG	1017	In Stock
50MG	1349	In Stock
100MG	1814	In Stock
200MG	Get Quote	In Stock
500MG	3618	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

Fluorobexarotene
Note

Research use only, not for human use.
Brief Description

Fluorobexarotene possesses an apparent RXR binding affinity that is 75% greater than Bexarotene.
Description

Fluorobexarotene (compound 20) is a potent retinoid-X-receptor (RXR) agonist, with a Ki value of 12 nM and an EC50 value of 43 nM for RXRα receptor. Fluorobexarotene possesses an apparent RXR binding affinity that is 75% greater than Bexarotene.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Metabolic Enzyme/Protease
Target

Retinoid Receptor
Recptor

Retinoid Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

1190848-23-7
Formula Weight

366.47
Molecular Formula

C24H27FO2
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 36 mg/mL (98.23 mM )
SMILES

CC1=CC2=C(C=C1C(=C)C1=CC(F)=C(C=C1)C(O)=O)C(C)(C)CCC2(C)C
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Wagner CE, et al. Modeling, synthesis and biological evaluation of potential retinoid X receptor (RXR) selective agonists: novel analogues of 4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydro-2-naphthyl)ethynyl]benzoic acid (bexarotene). J Med Chem. 2009 Oct?

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