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BX-517
CAS No. 850717-64-5
BX-517( BX-517 | BX 517 | BX517 | PDK1 inhibitor2 )
Catalog No. M17615 CAS No. 850717-64-5
BX-517 is a potent and selective inhibitor of PDK1.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 67 | In Stock |
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| 5MG | 61 | In Stock |
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| 10MG | 85 | In Stock |
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| 25MG | 147 | In Stock |
|
| 50MG | 269 | In Stock |
|
| 100MG | 423 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBX-517
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NoteResearch use only, not for human use.
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Brief DescriptionBX-517 is a potent and selective inhibitor of PDK1.
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DescriptionBX-517, also known as PDK1 inhibitor2, is a potent and selective PDK1 inhibitor.
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In Vitro——
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In Vivo——
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SynonymsBX-517 | BX 517 | BX517 | PDK1 inhibitor2
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PathwayMetabolic Enzyme/Protease
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TargetRetinoid Receptor
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RecptorPDK1
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number850717-64-5
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Formula Weight282.3
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Molecular FormulaC15H14N4O2
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 27 mg/mL; 95.64 mM
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SMILESO=C(Nc1cc2c(NC(=O)/C/2=C(\c2ccc[nH]2)/C)cc1)N
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Chemical Name(Z)-N-(3-(1-(1H-pyrrol-2-yl)ethylidene)-2-hydroxy-3H-indol-5-yl)carbamimidic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Islam I, et al. Indolinone based phosphoinositide-dependent kinase-1 (PDK1) inhibitors. Part 2: optimization of BX-517. Bioorg Med Chem Lett. 2007 Jul 15;17(14):3819-25.
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