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11β-HSD1-IN-1

CAS No. 1203956-47-1

11β-HSD1-IN-1( —— )

Catalog No. M32755 CAS No. 1203956-47-1

11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1, IC50: 52 nM) used for the treatment of pain.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	115	In Stock
5MG	107	In Stock
10MG	158	In Stock
25MG	236	In Stock
50MG	324	In Stock
100MG	442	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

11β-HSD1-IN-1
Note

Research use only, not for human use.
Brief Description

11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1, IC50: 52 nM) used for the treatment of pain.
Description

11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1), with an IC50 of 52 nM, and used for the treatment of pain.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Metabolic Enzyme/Protease
Target

Dehydrogenase
Recptor

Dehydrogenase
Research Area

——
Indication

——

Chemical Information

CAS Number

1203956-47-1
Formula Weight

399.77
Molecular Formula

C18H14ClF4N3O
Purity

>98% (HPLC)
Solubility

——
SMILES

CN1C(=NN=C1C(OC2=C(F)C=C(F)C=C2F)(C)C)C3=C(Cl)C=C(F)C=C3
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. THERAPEUTIC AGENT FOR PAIN. WO2012033070A1

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