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Calcium channel-modulator-1

CAS No. 136941-70-3

Calcium channel-modulator-1( —— )

Catalog No. M32746 CAS No. 136941-70-3

Calcium channel-modulator-1, a calcium channel-modulator (IC50: 0.8 μM), specializes in blocking aortic constriction.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 332 In Stock
5MG 258 In Stock
10MG 416 In Stock
25MG 708 In Stock
50MG 918 In Stock
100MG 1293 In Stock
200MG 1739 In Stock
500MG Get Quote In Stock
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Biological Information

  • Product Name
    Calcium channel-modulator-1
  • Note
    Research use only, not for human use.
  • Brief Description
    Calcium channel-modulator-1, a calcium channel-modulator (IC50: 0.8 μM), specializes in blocking aortic constriction.
  • Description
    Calcium channel-modulator-1 is a calcium channel modulator; blocks aortic contraction with an IC50 of 0.8 μM.
  • In Vitro
    ——
  • In Vivo
    Oral administration of Calcium channel-modulator-1 (20 mg/kg) causes a 35-37% decrease in systolic blood pressure in spontaneously hypertensive rats. However, iv administration of Calcium channel-modulator-1 to anesthetized spontaneously hypertensive rats causes a decrease in blood pressure which was more pronounced and long-lasting than that of nifedipine.
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Calcium Channel
  • Recptor
    Calcium Channel
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    136941-70-3
  • Formula Weight
    579.45
  • Molecular Formula
    C26H24Cl2N2O7S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C(OCCCN1S(=O)(=O)C=2C(C1=O)=CC=CC2)(=O)C=3C(C(C(OC)=O)=C(C)NC3C)C4=C(Cl)C(Cl)=CC=C4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Sunkel CE, et al. Synthesis of 3-[(2,3-dihydro-1,1,3-trioxo-1,2-benzisothiazol-2-yl)alkyl] 1,4-dihydropyridine-3,5-dicarboxylate derivatives as calcium channel modulators. J Med Chem. 1992 Jun 26;35(13):2407-14.?
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