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ARV-471
CAS No. 2229711-68-4
ARV-471( —— )
Catalog No. M28234 CAS No. 2229711-68-4
ARV-471 is a best-in-class, orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 851 | In Stock |
|
| 5MG | 437 | In Stock |
|
| 10MG | 622 | In Stock |
|
| 25MG | 924 | In Stock |
|
| 50MG | 1230 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameARV-471
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NoteResearch use only, not for human use.
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Brief DescriptionARV-471 is a best-in-class, orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
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DescriptionARV-471 is a best-in-class, orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetEstrogen Receptor/ERR
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RecptornAChR
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Research Area——
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Indication——
Chemical Information
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CAS Number2229711-68-4
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Formula Weight723.9
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Molecular FormulaC45H49N5O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 110 mg/mL (151.95 mM)
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SMILESOc1cc(CC[C@@H]([C@@H]2c(cc3)ccc3N3CCC(CN(CC4)CCN4c(cc4)cc(CN5[C@@H](CCC(N6)=O)C6=O)c4C5=O)CC3)c3ccccc3)c2cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Matthew J. Cheesman . Oceania: Antidepressant Medicinal Plants. Herbal Medicine in Depression. 2016, 483-527.
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