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Nitrocaramiphen hydrochloride
CAS No. 98636-73-8
Nitrocaramiphen hydrochloride( —— )
Catalog No. M27669 CAS No. 98636-73-8
Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 29 | In Stock |
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| 10MG | 46 | In Stock |
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| 25MG | 91 | In Stock |
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| 50MG | 145 | In Stock |
|
| 100MG | 214 | In Stock |
|
| 200MG | 306 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameNitrocaramiphen hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionNitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.
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DescriptionNitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.(In Vitro):Nitrocaramiphen hydrochloride binds with high affinity for M1 sites (Ki = 5.5 nM) and with a 71-fold selectivity over M2, and a 10-fold selectivity for the M1 over the M3 subtype.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetAChR
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RecptorTubulin polymerization
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Research Area——
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Indication——
Chemical Information
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CAS Number98636-73-8
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Formula Weight370.87
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Molecular FormulaC18H27ClN2O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 10 mg/mL (26.96 mM)
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SMILESCl.CCN(CC)CCOC(=O)C1(CCCC1)c1ccc(cc1)[N+]([O-])=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.R De Vincenzo, et al. Antiproliferative Activity of Colchicine Analogues on MDR-positive and MDR-negative Human Cancer Cell Lines. Anticancer Drug Des. 1998 Jan;13(1):19-33.
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