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BRL 52537 hydrochloride

CAS No. 112282-24-3

BRL 52537 hydrochloride( —— )

Catalog No. M27458 CAS No. 112282-24-3

BRL 52537 hydrochloride is a selective and specific KOR agonist which has been implicated in neuroprotection from ischemic neuronal injury.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 106 In Stock
5MG 156 In Stock
10MG 222 In Stock
25MG 413 In Stock
50MG 606 In Stock
100MG 862 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    BRL 52537 hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    BRL 52537 hydrochloride is a selective and specific KOR agonist which has been implicated in neuroprotection from ischemic neuronal injury.
  • Description
    BRL 52537 hydrochloride is a selective and specific KOR agonist which has been implicated in neuroprotection from ischemic neuronal injury. It is used for research into potential treatments for stroke and heart attack as well as more general brain research.(In Vivo):In rats treated with BRL 52537 during ischemia and early reperfusion, infarct volume was significantly attenuated in cortex and in caudoputamen.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    Opioid Receptor
  • Recptor
    RARγ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    112282-24-3
  • Formula Weight
    391.76
  • Molecular Formula
    C18H25Cl3N2O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(Cc(cc1)cc(Cl)c1Cl)N1C(CN2CCCC2)CCCC1.Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Hughes NE, et al. Identification of potent and selective retinoic acid receptor gamma (RARγ) antagonists for the treatment of osteoarthritis pain using structure based drug design. Bioorg Med Chem Lett. 2016 Jul 15;26(14):3274-3277.
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