LY2979165

CAS No. 1311385-32-6

LY2979165( mGlu2 agonist )

Catalog No. M26747 CAS No. 1311385-32-6

LY2979165 is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 113 In Stock
5MG 178 In Stock
10MG 237 In Stock
25MG 420 In Stock
50MG 617 In Stock
100MG 878 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    LY2979165
  • Note
    Research use only, not for human use.
  • Brief Description
    LY2979165 is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.
  • Description
    LY2979165 is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.(In Vivo):LY2979165 reduces BOLD signal and increases plasma levels of 2812223 in vivo.
  • In Vitro
    ——
  • In Vivo
    LY2979165 attenuated the ketamine-evoked BOLD phMRI signal in vivo.
  • Synonyms
    mGlu2 agonist
  • Pathway
    Neuroscience
  • Target
    GluR
  • Recptor
    NK1| NK3
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1311385-32-6
  • Formula Weight
    390.42
  • Molecular Formula
    C13H22N6O6S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?H2O : ≥ 50 mg/mL (128.07 mM)D)
  • SMILES
    N.O.C[C@H](N)C(=O)N[C@]1(C[C@@H](Sc2ncn[nH]2)[C@H]2[C@@H]([C@@H]12)C(O)=O)C(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Pawsey S, et al. Elinzanetant (NT-814), a Neurokinin 1,3 Receptor Antagonist, Reduces Estradiol and Progesterone in Healthy Women. J Clin Endocrinol Metab. 2021 Jul 13;106(8):e3221-e3234.
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