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Selisistat R-enantiomer
CAS No. 848193-69-1
Selisistat R-enantiomer( EX-527 (R-enantiomer) )
Catalog No. M26682 CAS No. 848193-69-1
Selisistat R-enantiomer is a SIRT1 inhibitor with much less activity than the R-enantiomer of Selisistat (IC50 of SIRT1 > 100 μM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 177 | Get Quote |
|
| 5MG | 314 | Get Quote |
|
| 10MG | 447 | Get Quote |
|
| 25MG | 714 | Get Quote |
|
| 50MG | 1017 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameSelisistat R-enantiomer
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NoteResearch use only, not for human use.
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Brief DescriptionSelisistat R-enantiomer is a SIRT1 inhibitor with much less activity than the R-enantiomer of Selisistat (IC50 of SIRT1 > 100 μM).
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DescriptionSelisistat R-enantiomer is a SIRT1 inhibitor with much less activity than the R-enantiomer of Selisistat (IC50 of SIRT1 > 100 μM).
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In Vitro——
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In Vivo——
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SynonymsEX-527 (R-enantiomer)
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PathwayChromatin/Epigenetic
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TargetSirtuin
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RecptorERK| hERG| IFN-γ| JNK| NF-κB| p38 MAPK| STAT| TLR
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Research Area——
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Indication——
Chemical Information
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CAS Number848193-69-1
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Formula Weight248.71
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Molecular FormulaC13H13ClN2O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (402.07 mM)
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SMILESNC(=O)[C@@H]1CCCc2c1[nH]c1ccc(Cl)cc21
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Liu XQ, et al. [Thymopolypeptides combined with matrine type alkaloids suppress HBV replication]. Zhongguo Zhong Yao Za Zhi. 2016 Apr;41(7):1275-1281. Chinese.
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