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N-Desmethyl-Apalutamide
CAS No. 1332391-11-3
N-Desmethyl-Apalutamide( N-Desmethyl Apalutamide )
Catalog No. M26314 CAS No. 1332391-11-3
N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 278 | In Stock |
|
| 5MG | 259 | In Stock |
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| 10MG | 373 | In Stock |
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| 25MG | 562 | In Stock |
|
| 50MG | 759 | In Stock |
|
| 100MG | 1014 | In Stock |
|
| 200MG | 1376 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameN-Desmethyl-Apalutamide
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NoteResearch use only, not for human use.
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Brief DescriptionN-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
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DescriptionN-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
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In Vitro——
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In Vivo——
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SynonymsN-Desmethyl Apalutamide
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PathwayMetabolic Enzyme/Protease
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TargetP450
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RecptorCYP2C9| HIV
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Research Area——
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Indication——
Chemical Information
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CAS Number1332391-11-3
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Formula Weight463.41
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Molecular FormulaC20H13F4N5O2S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (215.79 mM)
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SMILESNC(=O)c1ccc(cc1F)N1C(=S)N(C(=O)C11CCC1)c1cnc(C#N)c(c1)C(F)(F)F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Chen DF, et al. Anti-AIDS agents--XXVI. Structure-activity correlations of gomisin-G-related anti-HIV lignans from Kadsura interior and of related synthetic analogues. Bioorg Med Chem. 1997 Aug;5(8):1715-23.
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