Elinogrel
CAS No. 936500-94-6
Elinogrel( PRT060128 )
Catalog No. M26193 CAS No. 936500-94-6
Elinogrel is a competitive and reversible antagonist of platelet P2Y12 with IC50 of 20 nM and exhibits potent antiplatelet effects.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 115 | Get Quote |
|
| 10MG | 187 | Get Quote |
|
| 25MG | 376 | Get Quote |
|
| 50MG | 570 | Get Quote |
|
| 100MG | 795 | Get Quote |
|
| 500MG | 1647 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameElinogrel
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NoteResearch use only, not for human use.
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Brief DescriptionElinogrel is a competitive and reversible antagonist of platelet P2Y12 with IC50 of 20 nM and exhibits potent antiplatelet effects.
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DescriptionElinogrel is a competitive and reversible antagonist of platelet P2Y12 with IC50 of 20 nM and exhibits potent antiplatelet effects.
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In Vitro——
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In Vivo——
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SynonymsPRT060128
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PathwayGPCR/G Protein
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TargetP2Y Receptor
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RecptorNa+/Ca2+ Exchanger
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Research Area——
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Indication——
Chemical Information
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CAS Number936500-94-6
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Formula Weight523.94
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Molecular FormulaC20H15ClFN5O5S2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 62.5 mg/mL (119.29 mM)
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SMILESCNc1cc2[nH]c(=O)n(-c3ccc(NC(=O)NS(=O)(=O)c4ccc(Cl)s4)cc3)c(=O)c2cc1F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Chiesi M, et al. Structural dependency of the inhibitory action of benzodiazepines and related compounds on the mitochondrial Na+-Ca2+ exchanger. Biochem Pharmacol. 1988 Nov 15;37(22):4399-403.
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