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LSP-249

CAS No. 1801253-04-2

LSP-249( —— )

Catalog No. M23814 CAS No. 1801253-04-2

LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
2MG	36	In Stock
5MG	58	In Stock
10MG	87	In Stock
25MG	177	In Stock
50MG	295	In Stock
100MG	484	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

LSP-249
Note

Research use only, not for human use.
Brief Description

LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.
Description

LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

kallikrein
Research Area

——
Indication

——

Chemical Information

CAS Number

1801253-04-2
Formula Weight

431.92
Molecular Formula

C24H22ClN5O
Purity

>98% (HPLC)
Solubility

DMSO:31.25 mg/mL?(69.45 mM;?ultrasonic and warming and heat to 60°C)
SMILES

Cc1cc(N)nc(C)c1CNC(c1cc(Cc2ccc3ncc(Cl)cc3c2)ncc1)=O
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Andrew Mcdonald, et al. Therapeutic inhibitory compounds. Patent. WO2016011209A1.

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