DY-268
CAS No. 1609564-75-1
DY-268( —— )
Catalog No. M23707 CAS No. 1609564-75-1
DY-268 is a compound based on trisubstituted pyrazolamide without any FXR agonist activity and cytotoxicity and can be used as an effective FXR antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 85 | In Stock |
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| 5MG | 76 | In Stock |
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| 10MG | 122 | In Stock |
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| 25MG | 245 | In Stock |
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| 50MG | 445 | In Stock |
|
| 100MG | 641 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 1376 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDY-268
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NoteResearch use only, not for human use.
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Brief DescriptionDY-268 is a compound based on trisubstituted pyrazolamide without any FXR agonist activity and cytotoxicity and can be used as an effective FXR antagonist.
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DescriptionDY-268 is a compound based on trisubstituted pyrazolamide without any FXR agonist activity and cytotoxicity and can be used as an effective FXR antagonist (IC50 = 7.5 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetFXR
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RecptorFXR
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Research Area——
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Indication——
Chemical Information
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CAS Number1609564-75-1
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Formula Weight560.66
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Molecular FormulaC30H32N4O5S
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Purity>98% (HPLC)
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SolubilityDMSO:Soluble; Water: Insoluble
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SMILESCc(cc1)ccc1-c1nn(Cc2cc(OC)ccc2)cc1C(Nc1cc(S(N2CCOCC2)(=O)=O)c(C)cc1)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Roman-Lopez J, et al. Effect of the chemical impurities on the luminescence emission of natural apatites. Spectrochim Acta A Mol Biomol Spectrosc. 2014 May 21;126:142-7.
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