[Lys5,MeLeu9,Nle10]-NKA(4-10)( —— )

Catalog No. M22354 CAS No. 137565-28-7

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Product Name

[Lys5,MeLeu9,Nle10]-NKA(4-10)
Note

Research use only, not for human use.
Brief Description

Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
Description

Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
In Vitro

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In Vivo

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Synonyms

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Pathway

GPCR/G Protein
Target

Neurokinin Receptor
Recptor

NK2
Research Area

——
Indication

——

CAS Number

137565-28-7
Formula Weight

804
Molecular Formula

C39H65N9O9
Purity

>98% (HPLC)
Solubility

water:1 mg/mL
SMILES

CCCC[C@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CNC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](N)CC(O)=O)C(C)C)C(N)=O
Chemical Name

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1. Chassaing et al (1991) Selective agonists of NK-2 binding sites highly active on rat portal vein (NK-3 bioassay). Neuropeptides 19 91 PMID:

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