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Maropitant

CAS No. 147116-67-4

Maropitant( —— )

Catalog No. M20648 CAS No. 147116-67-4

Maropitant is a selective neurokinin (NK1) receptor antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 39 In Stock
5MG 65 In Stock
10MG 110 In Stock
25MG 177 In Stock
50MG 335 In Stock
100MG 500 In Stock
500MG 1098 In Stock
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Biological Information

  • Product Name
    Maropitant
  • Note
    Research use only, not for human use.
  • Brief Description
    Maropitant is a selective neurokinin (NK1) receptor antagonist.
  • Description
    Maropitant is a selective neurokinin (NK1) receptor antagonist.
  • In Vitro
    ——
  • In Vivo
    Treatment with 1 mg/kg Maropitant citrate, significantly reduces the size of ulcerative dermatitis (UD) lesions in mice. Intravenous Maropitant decreases MAC by 16%. In contrast, epidural administration of either saline or Maropitant does not change the MAC (2.17% and 1.92 %, respectively).
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Neurokinin Receptor
  • Recptor
    NK1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    147116-67-4
  • Formula Weight
    468.67
  • Molecular Formula
    C32H40N2O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:33.33 mg/mL (71.12 mM)
  • SMILES
    COc1ccc(cc1CN[C@H]1C2CCN(CC2)[C@H]1C(c1ccccc1)c1ccccc1)C(C)(C)C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Hickman M A Cox S R Mahabir S et al. Safety pharmacokinetics and use of the novel NK‐1 receptor antagonist maropitant (Cerenia TM ) for the prevention of emesis and motion sickness in cats[J]. Journal of Veterinary Pharmacology and Therapeutics 2008 31(3):220-229.
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