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AZ-33
CAS No. 1370290-34-8
AZ-33( AZ-33 | AZ 33 | AZ33 | LDHA Inhibitor 33 )
Catalog No. M17263 CAS No. 1370290-34-8
AZ-33 is an LDHA inhibitor. Binding affinity to 6-His-tagged human LDHA (2 to 322 amino acid residue) expressed in Escherichia coli BL21 (DE3) cells by SPR analysis with an active value of 0.093 μM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 92 | In Stock |
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| 10MG | 155 | In Stock |
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| 25MG | 302 | In Stock |
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| 50MG | 445 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameAZ-33
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NoteResearch use only, not for human use.
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Brief DescriptionAZ-33 is an LDHA inhibitor. Binding affinity to 6-His-tagged human LDHA (2 to 322 amino acid residue) expressed in Escherichia coli BL21 (DE3) cells by SPR analysis with an active value of 0.093 μM.
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DescriptionAZ-33, also known as LDHA Inhibitor 33, is a LDHA Inhibitor. Lactate dehydrogenase A (LDHA), a key enzyme involved in anaerobic glycolysis, is frequently deregulated in human malignancies.
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In Vitro——
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In Vivo——
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SynonymsAZ-33 | AZ 33 | AZ33 | LDHA Inhibitor 33
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PathwayNeuroscience
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TargetGluR
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RecptorLDHA
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Research Area——
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Indication——
Chemical Information
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CAS Number1370290-34-8
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Formula Weight497.56
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Molecular FormulaC25H27N3O6S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (200.98 mM)
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SMILESO=C(O)C(C(=O)O)Cc1ccc(cc1)CCCC(=O)NCCC(=O)Nc1ccc2c(c1)sc(n2)C
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Chemical Name2-(4-(4-((3-((2-Methylbenzo[d]thiazol-6-yl)amino)-3-oxopropyl)amino)-4-oxobutyl)benzyl)malonic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ward RA, et al.J Med Chem. 2012 Apr 12;55(7):3285-306.
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