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CAM4712
CAS No. ——
CAM4712( CAM 4712 | CAM-4712 )
Catalog No. M16980 CAS No. ——
CAM4712 (CAM-4712) is a potent and selective CK2α inhibitor with IC50 of 7 uM, exhibits cell growth inhibition in HCT116 cell line with IC50 of 10 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameCAM4712
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NoteResearch use only, not for human use.
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Brief DescriptionCAM4712 (CAM-4712) is a potent and selective CK2α inhibitor with IC50 of 7 uM, exhibits cell growth inhibition in HCT116 cell line with IC50 of 10 uM.
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DescriptionCAM4712 (CAM-4712) is a potent and selective CK2α inhibitor with IC50 of 7 uM, exhibits cell growth inhibition in HCT116 cell line with IC50 of 10 uM; displays good selectivity against the 20 closely related CMGC kinases; inhibits CK2α dependent phosphorylation of Ser129 of Akt1 in cellular assays, CAM4066 has numerous advantages over the previously reported CAM4066.
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In Vitro——
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In Vivo——
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SynonymsCAM 4712 | CAM-4712
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PathwayMetabolic Enzyme/Protease
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TargetCasein Kinase
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RecptorCasein Kinase
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight425.376
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Molecular FormulaC24H24Cl2N3+
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name2-(2-(((2,6-dichloro-2'-ethyl-[1,1'-biphenyl]-4-yl)methyl)amino)ethyl)-1H-benzo[d]imidazol-3-ium
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Iegre J, et al. Chem Sci. 2018 Feb 20;9(11):3041-3049.
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