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SirReal1
CAS No. 801227-82-7
SirReal1( SirReal 1 )
Catalog No. M15998 CAS No. 801227-82-7
A novel potent, selective Sirt2 inhibitor with IC50 of 3.745 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameSirReal1
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NoteResearch use only, not for human use.
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Brief DescriptionA novel potent, selective Sirt2 inhibitor with IC50 of 3.745 uM.
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DescriptionA novel potent, selective Sirt2 inhibitor with IC50 of 3.745 uM; displays no inhibitory activity against Sirt1 and Sirt 3 (IC50>100 uM).
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In Vitro——
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In Vivo——
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SynonymsSirReal 1
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PathwayChromatin/Epigenetic
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TargetSirtuin
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RecptorSirtuin
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Research Area——
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Indication——
Chemical Information
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CAS Number801227-82-7
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Formula Weight370.489
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Molecular FormulaC18H18N4OS2
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(NC1=NC=C(CC2=CC=CC=C2)S1)CSC3=NC(C)=CC(C)=N3
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Chemical NameN-(5-benzylthiazol-2-yl)-2-((4,6-dimethylpyrimidin-2-yl)thio)acetamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Schiedel M, et al. Angew Chem Int Ed Engl. 2016 Feb 5;55(6):2252-6.
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