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EHT 1864
CAS No. 754240-09-0
EHT 1864( —— )
Catalog No. M15867 CAS No. 754240-09-0
EHT 1864 is a potent Rac family GTPase inhibitor with Kd of 40 nM, 50 nM, 60 nM and 250 nM for Rac1, Rac1b, Rac2 and Rac3, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 98 | In Stock |
|
| 5MG | 76 | In Stock |
|
| 10MG | 124 | In Stock |
|
| 25MG | 200 | In Stock |
|
| 50MG | 375 | In Stock |
|
| 100MG | 565 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEHT 1864
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NoteResearch use only, not for human use.
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Brief DescriptionEHT 1864 is a potent Rac family GTPase inhibitor with Kd of 40 nM, 50 nM, 60 nM and 250 nM for Rac1, Rac1b, Rac2 and Rac3, respectively.
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DescriptionEHT 1864 is a potent Rac family GTPase inhibitor with Kd of 40 nM, 50 nM, 60 nM and 250 nM for Rac1, Rac1b, Rac2 and Rac3, respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetRho
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RecptorRac1| Rac1b| Rac2| Rac3
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number754240-09-0
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Formula Weight581.47
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Molecular FormulaC25H29Cl2F3N2O4S
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Purity>98% (HPLC)
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SolubilityDMSO:100 mg/mL warmed (171.97 mM); Ethanol:<1 mg/mL (<1 mM); Water:100 mg/mL (171.97 mM)
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SMILESFC(F)(F)C1=CC2=NC=CC(SCCCCCOC3=COC(CN4CCOCC4)=CC3=O)=C2C=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Shutes A, et al. J Biol Chem. 2007, 282(49), 35666-35678.
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