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Tiplaxtinin
CAS No. 393105-53-8
Tiplaxtinin( PAI-039 )
Catalog No. M14351 CAS No. 393105-53-8
Tiplaxtinin(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 63 | In Stock |
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| 2MG | 35 | In Stock |
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| 5MG | 56 | In Stock |
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| 10MG | 83 | In Stock |
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| 25MG | 148 | In Stock |
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| 50MG | 254 | In Stock |
|
| 100MG | 500 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 1070 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTiplaxtinin
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NoteResearch use only, not for human use.
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Brief DescriptionTiplaxtinin(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.
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DescriptionTiplaxtinin(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.
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In Vitro——
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In Vivo——
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SynonymsPAI-039
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PathwayMetabolic Enzyme/Protease
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TargetPAI-1
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RecptorPAI-1
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Research AreaMetabolic Disease
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Indication——
Chemical Information
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CAS Number393105-53-8
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Formula Weight439.38
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Molecular FormulaC24H16F3NO4
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Purity>98% (HPLC)
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SolubilityDMSO: 10 mM
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SMILESO=C(O)C(C1=CN(CC2=CC=CC=C2)C3=C1C=C(C4=CC=C(OC(F)(F)F)C=C4)C=C3)=O
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Chemical Name2-(1-benzyl-5-(4-(trifluoromethoxy)phenyl)-1H-indol-3-yl)-2-oxoacetic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Elokdah H, et al. J Med Chem. 2004 Jul 1;47(14):3491-4.
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